What is Tamoxifen?

Tamoxifen is a drug classified under the Selective Estrogen Receptor Modulator (SERMS). It is popularly known as Nolvadex and acts by selectively antagonizing the estrogen effect in some tissues like the breast tissue. Therefore, the use of SERMS in the treatment of breast cancer and Post Cycle Therapy in bodybuilders is to prevent enlargement of the breast tissue. SERMS in PCT therapy acts by stimulating the production of luteinizing hormone from the pituitary gland, which in turn stimulates the production of testosterone. The testosterone produced counteracts the low levels of testosterone brought about by the use of anabolic steroids in bodybuilders.

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Role of SERMS in an anabolic steroid cycle.

SERMS is added as a Post Cycle Therapy, which is after the successful 4-6 week anabolic steroid regimen. Since most anabolic steroids lower the level of testosterone, bodybuilders take Nolvadex to mitigate the effects of low testosterone, which are water retention and gynecomastia. It acts by inhibiting estrogen receptors in the pituitary gland, creating a false state of deficit of sex hormones in the body. As a result, the body produces gonadotropins, primarily the luteinizing hormone, which stimulates testosterone production, raising the levels of testosterone.

SERMS Vs Aromatase Inhibitors.

In some instances, the use of SERMS may not be adequate to mitigate the effect of anabolics. Hence, additional use of aromatase inhibitors may be beneficial. Aromatase inhibitors act by limiting the activity of the aromatase enzyme that is responsible for the conversion of testosterone to estrogen. Hence, the levels of testosterone are increased. The raised testosterone levels hinder breast development. AIs are effective in reducing the water-retention side effect of anabolics than SERMS. However, SERMS are more effective in the mitigation of gynecomastia.

SERMS for Gynecomastia.

Gynecomastia is a scientific term that refers to male breast development. Gynecomastia often occurs due to low testosterone levels caused by the use of anabolics. Nolvadex is used by bodybuilders to prevent gynecomastia associated with the use of anabolic steroids. SERMS acts by antagonizing the estrogen receptors in the breast tissue, thus prevent breast tissue development.

Tamoxifen PCT.

SERMS is used as a medication in Post Cycle Therapy to mitigate the effects of anabolic steroids in bodybuilders. It stimulates the production of testosterone naturally after a long period of its suppression due to anabolic use. However, it is not recommended for individuals who used progesterone-associated steroids as it would potentiate some harmful adverse effects.

Tamoxifen Dosage.

The recommended tamoxifen dosage after steroid therapy is 10-20 mg per day. However, if the steroids that one took are too strong to reverse its effect, the use of Nolvadex needs to be supplemented with AIs. When it is used in conjunction with PCT, the recommended dose is 40 mg for the initial half phase, followed by 20 mg in the last half period. AIs can be bought alongside SERMS from a tamoxifen shop.

Tamoxifen Side Effects.

Use of SERMS in women is associated with nausea, hot flashes, abnormal vaginal bleeding, dizziness, fatigue, and mood swings. In men tamoxifen side effects are low libido, headache, nausea, and vomiting. Where one wants to minimize the chances of experiencing Tamoxifen side effects, individuals are advised that individuals stick to the recommended dosages for SERMS. Acne is also a common Tamoxifen side effect associated with SERMS use.

Common Q n A about SERMS.

Some of the frequently asked questions about the use of SERMS in bodybuilders are:
1. Does Nolvadex cause an increase in testosterone levels?
Yes, it has an indirect effect on the levels of testosterone by stimulating the production of luteinizing hormone in the pituitary glands
2. Will SERMS cause weight gain?
Ideally, SERMS does not cause weight gain. However, the use of Nolvadex is associated with increased testosterone levels, which, in turn, increases the body’s lean muscle. Thus, SERMS use is associated with weight gain.
3. What are the benefits of tamoxifen PCT to bodybuilders?
SERMS are used to avert the low testosterone effect associated with anabolic steroids use. Therefore, tamoxifen use will halt breast formation in males who use steroids.
4. Where can one buy tamoxifen?
Nolvadex is a prescription medicine. one can buy tamoxifen from the local pharmacy or other tamoxifen shop.
Trusted Brands of Tamoxifen in the market are: